SCHEMBL29635217

SCHEMBL29635217

N#Cc1[nH]c2ccccc2c1C#N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 6/20 0.49
ALDH1A1 P00352 4/20 0.46
GPR3 P46089 1/20 0.46
HSD17B10 Q99714 1/20 0.46
DRD2 P14416 1/20 0.44
DRD4 P21917 1/20 0.44
DRD3 P35462 1/20 0.44
PDE1C Q14123 1/20 0.44
KDM4E B2RXH2 3/20 0.43
KMT2A Q03164 2/20 0.43
GAA P10253 2/20 0.43
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
CACNA1B Q00975 1/20 0.43
APBA1 Q02410 1/20 0.43
EGFR P00533 2/20 0.43
SRC P12931 1/20 0.43
GABRP O00591 1/20 0.43
GABRD O14764 1/20 0.43
GABRA1 P14867 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2464667 1.00 PDE9A (0.49) PDE9AALDH1A1GPR3HSD17B10DRD2
SCHEMBL3676401 0.79 AHR (0.57) PDE9AALDH1A1GPR3HSD17B10PDE1C
SCHEMBL16156592 0.78 ALDH1A1 (0.44) PDE9AALDH1A1GPR3HSD17B10DRD2
SCHEMBL8588245 0.78 ALDH1A1 (0.50) ALDH1A1GPR3HSD17B10DRD2DRD4
SCHEMBL20505152 0.78 ALDH1A1 (0.44) PDE9AALDH1A1GPR3HSD17B10DRD2
SCHEMBL9034264 0.78 ALDH1A1 (0.44) PDE9AALDH1A1GPR3HSD17B10DRD2
SCHEMBL2731190 0.78 DRD2 (0.47) PDE9AALDH1A1GPR3HSD17B10DRD2
SCHEMBL3680016 0.78 AHR (0.55) PDE9AALDH1A1GPR3HSD17B10DRD2
SCHEMBL1514832 0.78 PDE9A (0.47) PDE9AALDH1A1GPR3HSD17B10PDE1C
SCHEMBL5858501 0.78 PLA2G1B (0.59) PDE9AALDH1A1GPR3HSD17B10PDE1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114671880-B Synthesis and application of indole-2, 3-dinitrile antitumor compounds containing fatty amino 大连理工大学 2023-06-06 CN claimed
CN-114671880-A Synthesis and application of indole-2, 3-dinitrile antitumor compound containing aliphatic amino 大连理工大学 2022-06-28 CN claimed
CN-114671880-B Synthesis and application of indole-2, 3-dinitrile antitumor compounds containing fatty amino 大连理工大学 2023-06-06 CN disclosed
CN-114671880-B Synthesis and application of indole-2, 3-dinitrile antitumor compounds containing fatty amino 大连理工大学 2023-06-06 CN disclosed
CN-114671880-B Synthesis and application of indole-2, 3-dinitrile antitumor compounds containing fatty amino 大连理工大学 2023-06-06 CN disclosed
CN-114671880-A Synthesis and application of indole-2, 3-dinitrile antitumor compound containing aliphatic amino 大连理工大学 2022-06-28 CN disclosed
CN-114671880-A Synthesis and application of indole-2, 3-dinitrile antitumor compound containing aliphatic amino 大连理工大学 2022-06-28 CN disclosed
CN-114671880-A Synthesis and application of indole-2, 3-dinitrile antitumor compound containing aliphatic amino 大连理工大学 2022-06-28 CN disclosed