SCHEMBL29636711

SCHEMBL29636711

NCCC(N)c1cc(-c2ccc3ncccc3c2)nc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
POLB P06746 1/20 0.46
RAB9A P51151 1/20 0.46
SYK P43405 11/20 0.43
DYRK1A Q13627 1/20 0.42
ATR Q13535 1/20 0.42
GRM4 Q14833 1/20 0.40
AKT1 P31749 1/20 0.39
PRKCH P24723 1/20 0.39
PRKCE Q02156 1/20 0.39
TOP1 P11387 1/20 0.39
TXK P42681 1/20 0.39
KARS1 Q15046 1/20 0.39
SLK Q9H2G2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28967193 0.76 ALDH1A1 (0.59) SYK
Hydrochloric Acid SCHEMBL29636779 0.75 ALDH1A1 (0.57) SYK
SCHEMBL30261191 0.75 SYK (0.57) SYK
SCHEMBL23029627 0.75 SYK (0.57) SYK
SCHEMBL29875350 0.75 NPC1 (0.56) NPC1POLBRAB9ADYRK1AATR
SCHEMBL23015154 0.75 NPC1 (0.56) NPC1POLBRAB9ADYRK1AATR
SCHEMBL29636719 0.74 ALDH1A1 (0.49) NPC1RAB9ASYK
SCHEMBL23015344 0.72 GRM2 (0.46)
SCHEMBL29636726 0.72 GRM2 (0.46)
SCHEMBL30853278 0.71 ALDH1A1 (0.50) NPC1POLBRAB9ADYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4017492-A1 MOLECULES THAT BIND TO TDP-43 FOR THE TREATMENT OF AMYOTROPHIC LATERAL SCLEROSIS AND RELATED DISORDERS Biohaven Therapeutics Ltd. (US) 2022-06-29 EP claimed
WO-2024054807-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS AND TDP-43 MODULATORS BIOHAVEN THERAPEUTICS LTD. (VG) 2024-03-14 WO disclosed