SCHEMBL29639579

SCHEMBL29639579

O=C(NCc1cccc(C(F)(F)F)c1-c1cccc(CO)c1)OCC1c2ccccc2-c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.41
KMT2A Q03164 3/20 0.40
EPHX1 P07099 2/20 0.38
CHRM3 P20309 1/20 0.38
P2RX7 Q99572 2/20 0.37
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
OPRD1 P41143 1/20 0.37
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
FFAR1 O14842 1/20 0.36
MEN1 O00255 1/20 0.36
ATM Q13315 1/20 0.36
MDM2 Q00987 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30466820 0.86 EPHX2 (0.40) EPHX2KMT2AP2RX7KDM4ELMNA
SCHEMBL20530632 0.86 EPHX2 (0.40) EPHX2KMT2AP2RX7KDM4ELMNA
SCHEMBL29639583 0.86 EPHX1 (0.43) EPHX2KMT2AEPHX1CHRM3OPRD1
SCHEMBL20530666 0.86 RBP4 (0.41) EPHX2KMT2AP2RX7NR1H2NR1H3
SCHEMBL20530627 0.85 EPHX2 (0.47) EPHX2KMT2AEPHX1CHRM3OPRD1
SCHEMBL20530673 0.84 KMT2A (0.42) EPHX2KMT2ACHRM3OPRD1MEN1
SCHEMBL20530641 0.84 PTGDR2 (0.45) EPHX2KMT2ACHRM3OPRD1MEN1
SCHEMBL20530650 0.80 KMT2A (0.47) EPHX2KMT2AP2RX7OPRD1KDM4E
SCHEMBL18688054 0.79 EPHX2 (0.53) EPHX2KMT2AEPHX1CHRM3OPRD1
SCHEMBL20530629 0.79 CHRM3 (0.45) EPHX2KMT2AEPHX1CHRM3MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609905-B1 PEPTIDE MACROCYCLES AND USE THEREOF IN THE TREATMENT OF BACTERIAL INFECTIONS HOFFMANN LA ROCHE (CH) 2022-06-08 EP disclosed