SCHEMBL29640086

SCHEMBL29640086

NC(=O)N1Cc2nccnc2C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 7/20 0.40
HDAC1 Q13547 6/20 0.39
DPP8 Q6V1X1 1/20 0.35
DPP9 Q86TI2 1/20 0.35
ADORA3 P0DMS8 1/20 0.34
TSHR P16473 1/20 0.34
MC4R P32245 1/20 0.34
ADRA1A P35348 1/20 0.34
MC3R P41968 1/20 0.34
PARP1 P09874 1/20 0.32
CDK1 P06493 1/20 0.31
MYT1 Q01538 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CCNA2 P20248 1/20 0.30
CDK2 P24941 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27923200 0.79 DPP8 (0.57) DPP8DPP9
SCHEMBL28625656 0.72 NAMPT (0.37) PARP1CCNA2CDK2CCNA1
SCHEMBL22224502 0.72 DPP8 (0.44) HDAC2HDAC1DPP8DPP9TSHR
SCHEMBL28411097 0.72 DPP8 (0.39) DPP8DPP9TSHRPARP1ALDH1A1
SCHEMBL4753809 0.68 DPP8 (0.47) DPP8DPP9TSHRALDH1A1HTT
SCHEMBL31348202 0.67 HDAC1 (0.44) HDAC2HDAC1DPP8DPP9ALDH1A1
SCHEMBL30456600 0.67
SCHEMBL6120302 0.66 HDAC2 (0.49) HDAC2HDAC1
SCHEMBL29690628 0.66 HDAC2 (0.49) HDAC2HDAC1
SCHEMBL14738035 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114450271-B Ureas, amino and substituted heteroaryl compounds for Cbl-b inhibition 纽力克斯治疗公司 2024-09-20 CN disclosed
CN-114450271-A Ureas, amino and substituted heteroaryl compounds for Cbl-b inhibition 纽力克斯治疗公司 2022-05-06 CN disclosed