SCHEMBL29640629

SCHEMBL29640629

CC1(C)COc2cc(Br)ccc2C1N

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 5/20 0.36
KDM1B Q8NB78 1/20 0.36
ADRA2A P08913 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
BLM P54132 1/20 0.35
CHRNA1 P02708 1/20 0.34
CHRNG P07510 1/20 0.34
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
SLC6A2 P23975 1/20 0.34
CHRNB4 P30926 1/20 0.34
SLC6A4 P31645 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
SLC6A3 Q01959 1/20 0.34
CHRND Q07001 1/20 0.34
TMEM97 Q5BJF2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23362524 1.00 KDM1A (0.36) KDM1AKDM1BADRA2ALMNAMAPT
SCHEMBL3457236 0.81 TMEM97 (0.37) ADRA2ALMNAMAPTHTTBLM
SCHEMBL29640648 0.75 KDM1A (0.43) KDM1AKDM1B
SCHEMBL23362293 0.75 KDM1A (0.43) KDM1AKDM1B
SCHEMBL28768384 0.75 KDM4C (0.33)
SCHEMBL23362302 0.73 HTR2C (0.40)
SCHEMBL23363148 0.73 KDM4C (0.38) HTTTMEM97
SCHEMBL3456675 0.72 ADRA2A (0.35) ADRA2A
SCHEMBL31490434 0.71 KDM1A (0.44) KDM1AKDM1BADRA2ASLC6A2SLC6A4
SCHEMBL31490277 0.71 KDM1A (0.44) KDM1AKDM1BADRA2ASLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114641477-A Novel compound having inhibitory activity against glucose ceramide synthase or pharmaceutically acceptable salt thereof, method for preparing same, and pharmaceutical composition comprising same 柳韩洋行 2022-06-17 CN disclosed