SCHEMBL29640648

SCHEMBL29640648

CC1(C)COc2cc(Br)c(F)cc2C1N

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 6/20 0.43
KDM1B Q8NB78 4/20 0.43
KCNH2 Q12809 2/20 0.41
BACE1 P56817 1/20 0.36
AKR1B1 P15121 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23362293 1.00 KDM1A (0.43) KDM1AKDM1BKCNH2BACE1AKR1B1
SCHEMBL29640596 0.79 HTR2C (0.40)
SCHEMBL23362302 0.79 HTR2C (0.40)
SCHEMBL28768381 0.76 SLC9A1 (0.36) KDM1AKDM1BKCNH2BACE1AKR1B1
SCHEMBL23362524 0.75 KDM1A (0.36) KDM1AKDM1B
SCHEMBL29640629 0.75 KDM1A (0.36) KDM1AKDM1B
SCHEMBL23363127 0.74 AKR1B1 (0.38) KDM1AKDM1BKCNH2AKR1B1
SCHEMBL20449182 0.70 KDM1A (0.45) KDM1AKDM1BKCNH2
SCHEMBL23362436 0.68 AKR1B1 (0.36) KDM1AKDM1BBACE1AKR1B1
SCHEMBL29640614 0.68 AKR1B1 (0.36) KDM1AKDM1BBACE1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114641477-A Novel compound having inhibitory activity against glucose ceramide synthase or pharmaceutically acceptable salt thereof, method for preparing same, and pharmaceutical composition comprising same 柳韩洋行 2022-06-17 CN disclosed