SCHEMBL29640657

SCHEMBL29640657

COc1ccc(OC(C)C#N)cc1Br

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.45
RECQL P46063 1/20 0.40
CYP1A2 P05177 3/20 0.40
CYP2C19 P33261 3/20 0.40
HPGD P15428 3/20 0.40
CYP2D6 P10635 2/20 0.40
MAPT P10636 2/20 0.39
ALOX12 P18054 1/20 0.39
GAA P10253 1/20 0.39
PKM P14618 1/20 0.39
MEN1 O00255 2/20 0.37
LMNA P02545 2/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
TUBB1 Q9H4B7 2/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10746306 0.86 CA12 (0.53) ALDH1A1CYP1A2CYP2C19HPGDMAPT
SCHEMBL31063385 0.80 ALDH1A1 (0.52) ALDH1A1RECQLCYP1A2CYP2C19HPGD
SCHEMBL3931086 0.80 ALDH1A1 (0.52) ALDH1A1RECQLCYP1A2CYP2C19HPGD
SCHEMBL5226607 0.76 CA1 (0.48) ALDH1A1CYP1A2HPGDMAPTGAA
SCHEMBL10667940 0.75 ALDH1A1 (0.42) ALDH1A1RECQLCYP1A2CYP2C19HPGD
SCHEMBL29634588 0.73 CA12 (0.65) ALDH1A1CYP1A2CYP2C19HPGDCYP2D6
SCHEMBL258418 0.73 CA12 (0.65) ALDH1A1CYP1A2CYP2C19HPGDCYP2D6
Isopropylamine SCHEMBL28069314 0.73 HTR2A (0.56) ALDH1A1CYP2D6MAPTMEN1KMT2A
SCHEMBL5634995 0.72 CA12 (0.62) ALDH1A1CYP1A2CYP2C19HPGDCYP2D6
SCHEMBL4291308 0.71 ALDH1A1 (0.46) ALDH1A1RECQLCYP1A2CYP2C19HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114641477-B Compounds having inhibitory activity on glucosylceramide synthase or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-03-12 CN disclosed
CN-114641477-A Novel compound having inhibitory activity against glucose ceramide synthase or pharmaceutically acceptable salt thereof, method for preparing same, and pharmaceutical composition comprising same 柳韩洋行 2022-06-17 CN disclosed