SCHEMBL5634995

SCHEMBL5634995

COc1ccc(OC)c(Br)c1.[MgH2]

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.62
CA1 P00915 2/20 0.62
CA2 P00918 2/20 0.62
CA7 P43166 2/20 0.62
CA9 Q16790 2/20 0.62
CA14 Q9ULX7 2/20 0.62
ALDH1A1 P00352 4/20 0.54
MAPT P10636 3/20 0.54
MEN1 O00255 1/20 0.54
THRB P10828 1/20 0.54
KMT2A Q03164 1/20 0.54
CYP1A2 P05177 3/20 0.48
CYP1A1 P04798 2/20 0.48
CYP1B1 Q16678 2/20 0.48
CYP3A4 P08684 1/20 0.48
CTSL P07711 1/20 0.48
HTR2A P28223 2/20 0.47
HTR2C P28335 2/20 0.47
TUBB1 Q9H4B7 2/20 0.47
IDO1 P14902 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29634588 0.98 CA12 (0.65) CA12CA1CA2CA7CA9
SCHEMBL258418 0.98 CA12 (0.65) CA12CA1CA2CA7CA9
SCHEMBL9383598 0.89 CA12 (0.61) CA12CA1CA2CA7CA9
Isopropylamine SCHEMBL28069314 0.87 HTR2A (0.56) CA12CA1CA2CA7CA9
SCHEMBL38657587 0.86 ALDH1A1 (0.56) CA12CA1CA2CA7CA9
SCHEMBL31285028 0.85 CA12 (0.50) CA12CA1CA2CA7CA9
SCHEMBL31285041 0.85 CA12 (0.50) CA12CA1CA2CA7CA9
Propylamine SCHEMBL27607874 0.84 ADRA1A (0.56) CA12CA1CA2CA7CA9
SCHEMBL7403167 0.84 CA12 (0.60) CA12CA1CA2CA7CA9
Dimethylformamide SCHEMBL28323288 0.82 ALDH1A1 (0.49) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7297708-B2 Heteroaromatic substituted cyclopropane as corticotropin releasing hormone ligands BRISTOL-MYERS SQUIBB COMPANY (US) 2007-11-20 US disclosed
US-20030229091-A1 Heteroaromatic substituted cyclopropane as corticotropin releasing hormone ligands BRISTOL-MYERS SQUIBB COMPANY 2003-12-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030229091-A1 Heteroaromatic substituted cyclopropane as corticotropin releasing hormone ligands CRHR1, CRH, CRHR2 CA12 2779/4885CA1 1059/4885CA2 2868/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.