SCHEMBL29640758

SCHEMBL29640758

COc1ccc2c(c1)CN(c1nccc(-c3nccc(C#Cc4cc5ccccc5c(N)n4)n3)n1)C2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 8/20 0.41
ROCK1 Q13464 4/20 0.41
TUBB4A P04350 2/20 0.38
TUBB P07437 2/20 0.38
TUBA3C P0DPH7 2/20 0.38
TUBA1B P68363 2/20 0.38
TUBA4A P68366 2/20 0.38
TUBB4B P68371 2/20 0.38
TUBB3 Q13509 2/20 0.38
TUBB2A Q13885 2/20 0.38
TUBB8 Q3ZCM7 2/20 0.38
TUBA3E Q6PEY2 2/20 0.38
TUBA1A Q71U36 2/20 0.38
TUBA1C Q9BQE3 2/20 0.38
TUBB6 Q9BUF5 2/20 0.38
TUBB2B Q9BVA1 2/20 0.38
TUBB1 Q9H4B7 2/20 0.38
PDE10A Q9Y233 1/20 0.34
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29627697 0.86 ROCK2 (0.40) ROCK2ROCK1TUBB4ATUBBTUBA3C
SCHEMBL29640795 0.82 ROCK2 (0.42) ROCK2ROCK1PDE10AHCRTR1HCRTR2
SCHEMBL29627935 0.82 ROCK2 (0.52) ROCK2ROCK1PDE10AHCRTR1HCRTR2
SCHEMBL29640451 0.80 ROCK2 (0.44) ROCK2ROCK1
SCHEMBL29640938 0.80 ROCK2 (0.42) ROCK2ROCK1TUBB4ATUBBTUBA3C
SCHEMBL29640901 0.80 HCRTR1 (0.41) ROCK2ROCK1PDE10AHCRTR1HCRTR2
SCHEMBL29640913 0.79 ROCK2 (0.42) ROCK2ROCK1HCRTR1HCRTR2
SCHEMBL29627937 0.79 ROCK2 (0.54) ROCK2ROCK1
SCHEMBL29627955 0.78 ROCK2 (0.42) ROCK2ROCK1HCRTR1HCRTR2
SCHEMBL29627925 0.78 ROCK2 (0.43) ROCK2ROCK1HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed