SCHEMBL29640776

SCHEMBL29640776

O=c1ccnc(-c2ccncn2)n1Cl

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 11/20 0.37
CDC7 O00311 1/20 0.35
CCNT1 O60563 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CDK9 P50750 1/20 0.34
CCNA1 P78396 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
P2RX7 Q99572 3/20 0.33
GRM5 P41594 1/20 0.33
MAP4K4 O95819 1/20 0.33
EGFR P00533 1/20 0.33
FRK P42685 1/20 0.33
MAPK9 P45984 1/20 0.33
CSNK1A1 P48729 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29640916 0.72 SMN1; SMN2 (0.41) GSK3B
SCHEMBL29640865 0.71 GSK3B (0.36) GSK3BCDC7P2RX7GRM5
SCHEMBL10402322 0.68 HSP90AA1 (0.48) GSK3BCDC7CCNT1CCNA2CDK2
SCHEMBL2814353 0.67 HSP90AA1 (0.52) GSK3BCDC7CCNT1CCNA2CDK2
SCHEMBL30595872 0.67 HSP90AA1 (0.52) GSK3BCDC7CCNT1CCNA2CDK2
SCHEMBL4759558 0.66 GSK3B (0.55) GSK3B
SCHEMBL13910999 0.65 HSP90AA1 (0.50) GSK3BCDC7CCNT1CCNA2CDK2
SCHEMBL173216 0.62 GSK3B (0.61) GSK3B
SCHEMBL9903935 0.61 CYP2D6 (0.60) GSK3BGRM5MAP4K4EGFRFRK
SCHEMBL10841550 0.61 DYRK1A (0.57) GSK3BMAP4K4EGFRFRKMAPK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116209658-A Inhibitors of RHO-associated coiled coil kinase 安吉昂生物医药公司 2023-06-02 CN disclosed
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed