SCHEMBL29640865

SCHEMBL29640865

O=c1ccnc(-c2ccncn2)n1N1Cc2ccccc2C1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 13/20 0.36
P2RX7 Q99572 1/20 0.35
NAMPT P43490 2/20 0.34
CDC7 O00311 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
GRM5 P41594 1/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29640809 0.85 GSK3B (0.36) GSK3BCDC7CYP2D6
SCHEMBL6202952 0.73 GSK3B (0.40) GSK3BP2RX7NAMPTCDC7CYP2D6
SCHEMBL29640776 0.71 GSK3B (0.37) GSK3BP2RX7CDC7GRM5
SCHEMBL29640916 0.70 SMN1; SMN2 (0.41) GSK3BCYP2D6
SCHEMBL29640772 0.65 CYP1A2 (0.39) GSK3BNAMPTCYP2D6
SCHEMBL13742061 0.62 ALDH1A1 (0.54) ADORA3
SCHEMBL1569062 0.61 GSK3B (0.44) GSK3BCYP2D6
SCHEMBL10402322 0.61 HSP90AA1 (0.48) GSK3BP2RX7CDC7GRM5CYP2D6
SCHEMBL30595872 0.60 HSP90AA1 (0.52) GSK3BP2RX7CDC7GRM5CYP2D6
SCHEMBL2814353 0.60 HSP90AA1 (0.52) GSK3BP2RX7CDC7GRM5CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed