SCHEMBL29640808

SCHEMBL29640808

Cc1cn(-c2cccnc2N)cn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.50
CYP2A6 P11509 1/20 0.50
EGLN2 Q96KS0 1/20 0.46
NOS3 P29474 2/20 0.46
NOS2 P35228 2/20 0.46
NOS1 P29475 1/20 0.46
NR2E1 Q9Y466 1/20 0.38
PSEN1 P49768 4/20 0.37
PSEN2 P49810 4/20 0.37
APH1B Q8WW43 4/20 0.37
NCSTN Q92542 4/20 0.37
APH1A Q96BI3 4/20 0.37
PSENEN Q9NZ42 4/20 0.37
KCNH2 Q12809 3/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP19A1 P11511 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22199027 0.79 CYP2E1 (0.50) CYP2E1CYP2A6EGLN2PSEN1PSEN2
SCHEMBL17555719 0.79 NOS3 (0.46) CYP2E1CYP2A6EGLN2NOS3NOS2
SCHEMBL27819262 0.79 GAA (0.48) CYP2E1CYP2A6EGLN2NR2E1PSEN1
SCHEMBL12886318 0.76 CYP2E1 (0.42) CYP2E1CYP2A6EGLN2NR2E1PSEN1
SCHEMBL909404 0.76 PSEN1 (0.40) CYP2E1CYP2A6EGLN2NOS3NOS2
SCHEMBL909015 0.75 PSEN1 (0.43) CYP2E1CYP2A6EGLN2NR2E1PSEN1
SCHEMBL29949085 0.74 MAP3K5 (0.41) NOS3NOS2NOS1
SCHEMBL15633080 0.74 CYP2E1 (0.47) CYP2E1CYP2A6EGLN2PSEN1PSEN2
SCHEMBL16302917 0.74 GAA (0.50) NOS3NOS2NOS1AMY1AKDM4E
SCHEMBL27927385 0.72 HSP90AA1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112218857-B P300/CBP HAT inhibitors and methods of use thereof 星座制药公司 2023-11-21 CN disclosed
CN-114450005-A Compounds for the treatment of neurological disorders 星座制药公司 2022-05-06 CN disclosed