SCHEMBL22199027

SCHEMBL22199027

Cc1cn(-c2cccnc2Cl)cn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.50
CYP2A6 P11509 1/20 0.50
EGLN2 Q96KS0 1/20 0.46
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP19A1 P11511 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
PSEN1 P49768 7/20 0.36
PSEN2 P49810 7/20 0.36
APH1B Q8WW43 7/20 0.36
NCSTN Q92542 7/20 0.36
APH1A Q96BI3 7/20 0.36
PSENEN Q9NZ42 7/20 0.36
KCNH2 Q12809 1/20 0.34
PHF8 Q9UPP1 1/20 0.34
DOT1L Q8TEK3 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11569105 0.80 NOS3 (0.36) DOT1L
SCHEMBL29640808 0.79 CYP2E1 (0.50) CYP2E1CYP2A6EGLN2CYP1A2CYP3A4
SCHEMBL22185259 0.79 CPB1 (0.33) CYP2E1CYP2A6DOT1L
SCHEMBL22199076 0.79 PHF8 (0.51) CYP2E1CYP2A6EGLN2CYP1A2CYP3A4
SCHEMBL15633080 0.74 CYP2E1 (0.47) CYP2E1CYP2A6EGLN2CYP1A2CYP3A4
SCHEMBL951160 0.74 GAA (0.44) DOT1L
SCHEMBL27747138 0.71 CYP2E1 (0.45) CYP2E1CYP2A6EGLN2CYP1A2CYP3A4
SCHEMBL27159701 0.71 CYP1A2 (0.51) CYP2E1CYP2A6EGLN2CYP1A2CYP3A4
SCHEMBL27768055 0.71 CYP2E1 (0.45) CYP2E1CYP2A6EGLN2CYP1A2CYP3A4
SCHEMBL27417595 0.71 CYP2E1 (0.45) CYP2E1CYP2A6EGLN2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020141439-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-09 WO disclosed