SCHEMBL29640870

SCHEMBL29640870

C(#Cn1ncc2ccccc21)c1ccnc(-c2ccnc(N3CCC(c4ccccc4)CC3)n2)n1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.43
DYRK1A Q13627 12/20 0.38
DKK1 O94907 2/20 0.37
ROCK2 O75116 1/20 0.35
DHFR P00374 1/20 0.35
SCN9A Q15858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29640982 0.95 ROCK2 (0.42) ACACBDYRK1AROCK2SCN9A
SCHEMBL29640903 0.93 DYRK1A (0.38) ACACBDYRK1ADKK1
SCHEMBL29640965 0.88 DYRK1A (0.41) ACACBDYRK1AROCK2
SCHEMBL29640843 0.87 MAPT (0.40) DYRK1A
Trifluoroacetic Acid SCHEMBL29640829 0.84 ACACB (0.37) ACACBDYRK1A
SCHEMBL29640910 0.84 ROCK2 (0.48) ACACBDYRK1AROCK2
SCHEMBL29640817 0.84 DYRK1A (0.37) DYRK1ASCN9A
SCHEMBL29640810 0.82 DYRK1A (0.36) DYRK1AROCK2
SCHEMBL29640876 0.81 DYRK1A (0.37) DYRK1A
SCHEMBL29640867 0.81 CYP11B2 (0.38) DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed