Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL29640902

FC(F)(F)c1ccc2c(c1)CN(c1nccc(-c3nccc(C#Cn4ncc5ccccc54)n3)n1)C2.O=C(O)C(F)(F)F

nearest known ligand 0.37

Full drug profile on Sugi Atlas →

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.37
HCRTR2 O43614 2/20 0.37
NAMPT P43490 4/20 0.36
SCN9A Q15858 1/20 0.33
EIF2AK4 Q9P2K8 1/20 0.32
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
KDR P35968 1/20 0.30
CNR2 P34972 1/20 0.30
CRHR1 P34998 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29640778 0.84 ROCK2 (0.38) HCRTR1HCRTR2NAMPT
SCHEMBL29640810 0.84 DYRK1A (0.36)
Trifluoroacetic Acid SCHEMBL29640829 0.83 ACACB (0.37) HCRTR1HCRTR2
SCHEMBL29640878 0.83 DYRK1A (0.32) SCN9A
SCHEMBL29640938 0.81 ROCK2 (0.42) HCRTR1HCRTR2NAMPTSCN9A
SCHEMBL29640858 0.80 DYRK1A (0.33)
SCHEMBL29640949 0.79 MAP4K1 (0.37) KDR
Trifluoroacetic Acid SCHEMBL29640927 0.79 POLB (0.40)
SCHEMBL29640827 0.78 PDE10A (0.33) HCRTR1HCRTR2
SCHEMBL29640843 0.75 MAPT (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed