SCHEMBL29640878

SCHEMBL29640878

Brc1ccc2c(c1)CN(c1nccc(-c3nccc(C#Cn4ncc5ccccc54)n3)n1)C2

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 6/20 0.32
SCN9A Q15858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29640810 0.91 DYRK1A (0.36) DYRK1A
SCHEMBL29640778 0.89 ROCK2 (0.38) DYRK1A
SCHEMBL29640938 0.87 ROCK2 (0.42) SCN9A
SCHEMBL29640858 0.86 DYRK1A (0.33) DYRK1A
SCHEMBL29640949 0.85 MAP4K1 (0.37)
SCHEMBL29640812 0.83 TIPARP (0.39) SCN9A
SCHEMBL29640827 0.83 PDE10A (0.33) DYRK1A
Trifluoroacetic Acid SCHEMBL29640902 0.83 HCRTR1 (0.37) SCN9A
SCHEMBL29640839 0.81 DYRK1A (0.34) DYRK1A
SCHEMBL29640968 0.81 FAAH (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed