SCHEMBL29643035

SCHEMBL29643035

NC(=O)c1cnc2ccccc2c1N1CCOCC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
ALDH1A1 P00352 5/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
AURKA O14965 1/20 0.51
RPS6KB1 P23443 1/20 0.51
GRM5 P41594 1/20 0.49
PKM P14618 1/20 0.48
PTK2 Q05397 1/20 0.48
GAA P10253 2/20 0.47
MAPT P10636 1/20 0.47
TP53 P04637 2/20 0.46
KDM4E B2RXH2 2/20 0.45
HSD17B10 Q99714 2/20 0.45
GLA P06280 1/20 0.45
HPGD P15428 1/20 0.45
RAB9A P51151 1/20 0.45
LRRK2 Q5S007 1/20 0.45
USP2 O75604 1/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5093454 0.80 MEN1 (0.45) MEN1KMT2AALDH1A1SMN1; SMN2AURKA
SCHEMBL5096140 0.79 MEN1 (0.47) MEN1KMT2AALDH1A1SMN1; SMN2GRM5
SCHEMBL19989121 0.78 PIK3R2 (0.57)
SCHEMBL3830977 0.76 PTK2 (0.54) MEN1KMT2AALDH1A1SMN1; SMN2GRM5
SCHEMBL19988980 0.76 PIK3R2 (0.59) MEN1KMT2AALDH1A1SMN1; SMN2GAA
SCHEMBL19989078 0.76 PIK3C2B (0.56)
SCHEMBL29643198 0.75 RPS6KB1 (0.47) MEN1KMT2AALDH1A1SMN1; SMN2AURKA
SCHEMBL5093463 0.75 MEN1 (0.45) MEN1KMT2AALDH1A1SMN1; SMN2GRM5
SCHEMBL19989239 0.74 PIK3R2 (0.57) MEN1KMT2AALDH1A1SMN1; SMN2GAA
SCHEMBL30604174 0.74 PKM (0.81) MEN1KMT2AALDH1A1SMN1; SMN2AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4255911-A1 BICYCLIC DERIVATIVES Elanco Tiergesundheit AG (CH) 2023-10-11 EP claimed
WO-2022117783-A1 BICYCLIC DERIVATIVES ELANCO TIERGESUNDHEIT AG (CH) 2022-06-09 WO claimed
EP-4255911-A1 BICYCLIC DERIVATIVES Elanco Tiergesundheit AG (CH) 2023-10-11 EP disclosed
WO-2022117783-A1 BICYCLIC DERIVATIVES ELANCO TIERGESUNDHEIT AG (CH) 2022-06-09 WO disclosed