SCHEMBL29644341

SCHEMBL29644341

O=C(c1ccccc1)N1CCc2c(Br)cccc2C1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABHD6 Q9BV23 3/20 0.55
AKR1C3 P42330 1/20 0.53
HPGD P15428 6/20 0.52
ALDH1A1 P00352 3/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
TRAP1 Q12931 1/20 0.52
LMNA P02545 2/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CA7 P43166 1/20 0.51
CA9 Q16790 1/20 0.51
CA14 Q9ULX7 1/20 0.51
KDM4E B2RXH2 1/20 0.50
HTT P42858 1/20 0.49
NAMPT P43490 2/20 0.48
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
PTGS1 P23219 1/20 0.46
NPC1 O15118 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28739037 1.00 ABHD6 (0.55) ABHD6AKR1C3HPGDALDH1A1SMN1; SMN2
SCHEMBL1550147 0.85 ABHD6 (0.60) ABHD6AKR1C3SMN1; SMN2TRAP1NPC1
SCHEMBL29644313 0.84 CA1 (0.53) ABHD6HPGDALDH1A1SMN1; SMN2LMNA
SCHEMBL28739107 0.84 CA1 (0.53) ABHD6HPGDALDH1A1SMN1; SMN2LMNA
SCHEMBL3163275 0.84 HPGD (0.53) AKR1C3HPGDALDH1A1SMN1; SMN2LMNA
SCHEMBL29644426 0.83 HPGD (0.70) ABHD6HPGDALDH1A1SMN1; SMN2TRAP1
SCHEMBL28739023 0.83 HPGD (0.70) ABHD6HPGDALDH1A1SMN1; SMN2TRAP1
SCHEMBL10211721 0.83 HPGD (0.56) HPGDALDH1A1SMN1; SMN2TRAP1LMNA
SCHEMBL4008584 0.81 NOTUM (0.61) ABHD6AKR1C3TRAP1LMNA
SCHEMBL13051864 0.81 HPGD (0.50) HPGDALDH1A1SMN1; SMN2LMNACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114507181-B Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-03-26 CN disclosed
CN-114507181-A Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-05-17 CN disclosed