SCHEMBL29645523

SCHEMBL29645523

COc1cccc2c1nc(Nc1ccccnc1=O)n1nc(-c3cnn(C4CCC4)c3)nc21

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.36
PDE9A O76083 1/20 0.36
ADORA2A P29274 8/20 0.35
TP53 P04637 1/20 0.35
PAK1 Q13153 1/20 0.34
TNF P01375 3/20 0.34
LITAF Q99732 3/20 0.34
PIK3CA P42336 1/20 0.34
TTK P33981 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29646043 0.97 BRD4 (0.39) BRD4PDE9AADORA2ATP53PAK1
SCHEMBL29645911 0.88 CLK2 (0.33)
SCHEMBL29645614 0.88 TTK (0.39) BRD4ADORA2ATP53TTK
SCHEMBL29646004 0.86 MAPT (0.39) TP53
SCHEMBL29645561 0.85 MAP3K5 (0.34) PIK3CA
SCHEMBL29645641 0.84 TP53 (0.39) ADORA2ATP53TNFLITAFTTK
SCHEMBL29646080 0.82 MAPT (0.40) TP53
SCHEMBL29645741 0.81 KDM4E (0.48) ADORA2ATP53
SCHEMBL29645807 0.81 TP53 (0.39) TP53TTK
SCHEMBL22988377 0.81 ADORA2A (0.38) BRD4PDE9AADORA2APAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed