SCHEMBL29649401

SCHEMBL29649401

CS(=O)(=O)c1ccc2c(c1)CCCC2O

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 16/20 0.55
CYP3A4 P08684 1/20 0.44
IDO1 P14902 1/20 0.44
TDO2 P48775 1/20 0.44
PGR P06401 1/20 0.43
PNMT P11086 1/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29649410 0.88 HTR6 (0.46) HTR6CYP3A4IDO1TDO2PNMT
SCHEMBL7790505 0.86 CA12 (0.45) HTR6PGRCA12CA1CA2
SCHEMBL14009938 0.81 HTR6 (0.66) HTR6
SCHEMBL1282130 0.81 HTR6 (0.66) HTR6
SCHEMBL3184750 0.81 HTR6 (0.66) HTR6
SCHEMBL1003328 0.78 CYP3A4 (0.46) HTR6CYP3A4IDO1TDO2PNMT
SCHEMBL25081060 0.76 HTR6 (0.49) HTR6CYP3A4IDO1TDO2PNMT
SCHEMBL7909262 0.76 CA1 (0.47) HTR6PGRCA12CA1CA2
SCHEMBL17141459 0.76 SCN5A (0.44) HTR6CA12CA1CA2CA7
SCHEMBL17141458 0.76 SCN5A (0.44) HTR6CA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3394068-B1 TDO2 INHIBITORS GENENTECH INC (US) 2024-09-11 EP disclosed
CN-110072864-B TDO2 inhibitors 基因泰克公司 2022-05-27 CN disclosed