SCHEMBL29649948

SCHEMBL29649948

CC(C)(C)OC(=O)N(C(=O)OC(C)(C)C)c1nccc2cc(N)ccc12

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.36
NR1H4 Q96RI1 8/20 0.34
GRM4 Q14833 2/20 0.34
SYK P43405 1/20 0.34
NR1H2 P55055 1/20 0.33
SSTR4 P31391 1/20 0.32
PLAU P00749 1/20 0.32
GRM2 Q14416 1/20 0.32
AAK1 Q2M2I8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29508504 1.00 PDPK1 (0.36) PDPK1NR1H4GRM4SYKNR1H2
SCHEMBL1438293 1.00 PDPK1 (0.36) PDPK1NR1H4GRM4SYKNR1H2
SCHEMBL23012937 0.94 NR1H4 (0.35) PDPK1NR1H4GRM4SYKNR1H2
SCHEMBL27673955 0.89 NR1H4 (0.34) NR1H4GRM4NR1H2SSTR4PLAU
SCHEMBL2857004 0.86 NR1H4 (0.33) NR1H4GRM4NR1H2SSTR4PLAU
SCHEMBL29733555 0.86 AURKA (0.33)
SCHEMBL8233620 0.85 GABRG2 (0.39) PDPK1NR1H4GRM4SYKSSTR4
SCHEMBL22277233 0.84 NR1H4 (0.40) PDPK1NR1H4GRM2
SCHEMBL17221287 0.84 ROCK1 (0.47) PDPK1NR1H4NR1H2GRM2
SCHEMBL29481424 0.84 ROCK1 (0.47) PDPK1NR1H4NR1H2GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025049326-A1 TRICYCLIC HETEROAROMATIC INHIBITORS OF KLK5 BIOCRYST PHARMACEUTICALS, INC. (US) 2025-03-06 WO disclosed
EP-4255900-A2 ENZYME INHIBITORS Kalvista Pharmaceuticals Limited (GB) 2023-10-11 EP disclosed
US-20220298141-A1 ENZYME INHIBITORS KALVISTA PHARMACEUTICALS LIMITED (GB) 2022-09-22 US disclosed
EP-4017849-A1 ENZYME INHIBITORS Kalvista Pharmaceuticals Limited (GB) 2022-06-29 EP disclosed
WO-2022118016-A2 ENZYME INHIBITORS KALVISTA PHARMACEUTICALS LIMITED (GB) 2022-06-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220298141-A1 ENZYME INHIBITORS SERPINB1, ACE, GAA PDPK1 3344/4885NR1H4 545/4885GRM4 4592/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.