SCHEMBL29650608

SCHEMBL29650608

CC(C)(Nc1ncnc2cnccc12)C(F)(F)F

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
LATS1 O95835 16/20 0.60
LATS2 Q9NRM7 13/20 0.60
EGFR P00533 3/20 0.48
CYP1A2 P05177 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22302812 0.84 LATS1 (0.56) LATS1LATS2EGFRCYP1A2
SCHEMBL29650600 0.75 LATS1 (0.61) LATS1LATS2EGFR
SCHEMBL20574756 0.75 LATS1 (1.00) LATS1LATS2
SCHEMBL31375768 0.73 EGFR (0.65) LATS1EGFRCYP1A2
SCHEMBL3322882 0.73 EGFR (0.56) LATS1LATS2EGFR
SCHEMBL20574249 0.72 LATS1 (1.00) LATS1LATS2
SCHEMBL26177166 0.72 LATS1 (1.00) LATS1LATS2
SCHEMBL29650587 0.72 LATS1 (0.56) LATS1LATS2EGFR
SCHEMBL31375184 0.72 EGFR (0.53) LATS1EGFR
SCHEMBL20547766 0.71 LATS1 (1.00) LATS1LATS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114621222-A 6-6 fused bicyclic heteroaryl compounds and their use as LATS inhibitors 诺华股份有限公司 2022-06-14 CN claimed
CN-114703144-A 6-6 fused bicyclic heteroaryl compounds and their use as LATS inhibitors 诺华股份有限公司 2022-07-05 CN disclosed