SCHEMBL29655112

SCHEMBL29655112

O=C(O)c1ccc(Cc2ccc(F)c(Br)c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.47
RXRA P19793 2/20 0.47
RXRB P28702 2/20 0.47
RXRG P48443 1/20 0.47
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA9 Q16790 2/20 0.46
CA12 O43570 1/20 0.46
CA14 Q9ULX7 1/20 0.46
ALDH1A1 P00352 2/20 0.43
TSHR P16473 1/20 0.42
PTPN1 P18031 1/20 0.41
ERN1 O75460 1/20 0.41
VNN1 O95497 1/20 0.41
NR4A2 P43354 1/20 0.41
IDO1 P14902 1/20 0.40
TDO2 P48775 1/20 0.40
FAAH O00519 1/20 0.40
EGFR P00533 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28797926 1.00 SRD5A2 (0.47) SRD5A2RXRARXRBRXRGCA1
SCHEMBL1039881 0.80 CALM1 (0.48) CA1CA2CA9CA12CA14
SCHEMBL31302316 0.80 TTR (0.50) SRD5A2CA1CA2CA9CA12
SCHEMBL104151 0.80 TTR (0.50) SRD5A2CA1CA2CA9CA12
SCHEMBL3901537 0.78 KDM4E (0.45) ALDH1A1IDO1EGFR
Fluoride SCHEMBL11181401 0.78 TTR (0.48) SRD5A2CA1CA2CA9CA12
Bromide SCHEMBL11166294 0.78 TTR (0.48) SRD5A2CA1CA2CA9CA12
Hydrochloric Acid SCHEMBL6520005 0.78 TTR (0.48) SRD5A2CA1CA2CA9CA12
SCHEMBL27661360 0.78 KDM4E (0.62) SRD5A2RXRARXRBRXRGCA1
SCHEMBL68390 0.78 SRD5A2 (0.69) SRD5A2RXRARXRBRXRGCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843874-B Phthalazine derivatives useful as inhibitors of PARP1, PARP2 and/or tubulin for the treatment of cancer 加利福尼亚大学董事会 2022-05-27 CN disclosed