SCHEMBL29655290

SCHEMBL29655290

Cc1ccccc1-c1ccc(N)c([N+](=O)[O-])c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.64
MAPT P10636 3/20 0.64
MEN1 O00255 2/20 0.64
POLB P06746 2/20 0.64
KMT2A Q03164 2/20 0.64
TSHR P16473 3/20 0.56
ALDH1A1 P00352 4/20 0.50
CYP3A4 P08684 4/20 0.50
ALOX15 P16050 1/20 0.50
HSD17B10 Q99714 1/20 0.49
NPSR1 Q6W5P4 1/20 0.47
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
PKM P14618 1/20 0.44
LMNA P02545 1/20 0.44
RECQL P46063 1/20 0.44
HSP90AA1 P07900 1/20 0.43
CDK5 Q00535 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28258156 1.00 TDP1 (0.64) TDP1MAPTMEN1POLBKMT2A
O-Tolylamine SCHEMBL25436024 0.86 TDP1 (0.71) TDP1MAPTMEN1POLBKMT2A
SCHEMBL12117513 0.85 HSD17B10 (0.58) TDP1MAPTMEN1KMT2ATSHR
SCHEMBL3270267 0.84 S1PR1 (0.56) TDP1MAPTMEN1POLBKMT2A
SCHEMBL29655203 0.81 TDP1 (0.64) TDP1MAPTMEN1POLBKMT2A
SCHEMBL27864754 0.81 TDP1 (0.64) TDP1MAPTMEN1POLBKMT2A
SCHEMBL10714748 0.81 TDP1 (0.64) TDP1MAPTMEN1POLBKMT2A
SCHEMBL719169 0.81 TDP1 (0.64) TDP1MAPTMEN1POLBKMT2A
SCHEMBL29655079 0.81 TDP1 (0.64) TDP1MAPTMEN1POLBKMT2A
SCHEMBL6318909 0.81 ALDH1A1 (0.49) TDP1MAPTMEN1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843874-B Phthalazine derivatives useful as inhibitors of PARP1, PARP2 and/or tubulin for the treatment of cancer 加利福尼亚大学董事会 2022-05-27 CN disclosed