SCHEMBL29655508

SCHEMBL29655508

Nc1ncc(-c2ccc(C(F)(F)F)cc2)c(N)n1

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DHFR P00374 5/20 0.55
CDK5 Q00535 2/20 0.53
CDK5R1 Q15078 2/20 0.53
CLK1 P49759 2/20 0.49
ADORA2A P29274 1/20 0.48
ADORA1 P30542 1/20 0.48
HEXA P06865 1/20 0.48
HEXB P07686 1/20 0.48
MAP4K4 O95819 1/20 0.46
JAK2 O60674 1/20 0.46
KIF11 P52732 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1388289 1.00 DHFR (0.55) DHFRCDK5CDK5R1CLK1ADORA2A
SCHEMBL30584612 0.89 DHFR (0.49) DHFRCDK5CDK5R1CLK1ADORA2A
SCHEMBL1388479 0.83 ADORA2A (0.51) DHFRADORA2AADORA1
SCHEMBL29655536 0.81 ADORA2A (0.72) DHFRADORA2AADORA1
SCHEMBL1388662 0.81 ADORA2A (0.72) DHFRADORA2AADORA1
SCHEMBL4629601 0.80 ADORA1 (0.63) DHFRADORA2AADORA1MAP4K4
SCHEMBL30488033 0.80 ADORA1 (0.63) DHFRADORA2AADORA1MAP4K4
Hydrochloric Acid SCHEMBL27752359 0.80 ADORA2A (0.71) DHFRADORA2AADORA1
SCHEMBL31612551 0.80 DHFR (0.61) DHFRADORA2AADORA1
SCHEMBL29116207 0.80 DHFR (0.61) DHFRADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114621206-B 5-substituted pyrimidine diamine derivative and preparation method and application thereof 安徽医科大学 2023-11-24 CN disclosed
CN-116685583-A Pyrimidine compounds, compositions and pharmaceutical uses thereof 缆图药品公司 2023-09-01 CN disclosed
CN-114621206-A 5-substituted pyrimidinediamine derivative and preparation method and application thereof 安徽医科大学 2022-06-14 CN disclosed