SCHEMBL4629601

SCHEMBL4629601

Nc1ncc(-c2ccc(F)cc2)c(N)n1

nearest known ligand 0.68

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.63
DHFR P00374 7/20 0.57
P2RX3 P56373 1/20 0.47
P2RX2 Q9UBL9 1/20 0.47
TDO2 P48775 1/20 0.46
KMT2A Q03164 1/20 0.44
ADORA2A P29274 1/20 0.44
USP7 Q93009 1/20 0.43
CCNE1 P24864 1/20 0.42
CDK2 P24941 1/20 0.42
MAP4K4 O95819 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30488033 1.00 ADORA1 (0.63) ADORA1DHFRP2RX3P2RX2TDO2
SCHEMBL31612551 0.84 DHFR (0.61) ADORA1DHFRKMT2AADORA2A
SCHEMBL29116207 0.84 DHFR (0.61) ADORA1DHFRKMT2AADORA2A
SCHEMBL29913206 0.81 DHFR (0.67) DHFRTDO2KMT2AMAP4K4
SCHEMBL1936800 0.81 DHFR (0.57) ADORA1DHFRKMT2AADORA2A
SCHEMBL736022 0.81 DHFR (0.58) ADORA1DHFRKMT2AADORA2AUSP7
SCHEMBL4613214 0.81 DHFR (0.53) ADORA1DHFR
SCHEMBL1388506 0.81 DHFR (0.67) DHFRTDO2KMT2AMAP4K4
SCHEMBL29655508 0.80 DHFR (0.55) ADORA1DHFRADORA2AMAP4K4
SCHEMBL1388289 0.80 DHFR (0.55) ADORA1DHFRADORA2AMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012115479-A2 DIAMINOPYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 2012-08-30 WO claimed
CN-113061116-A Aminopyrimidine compound, preparation method, composition and application thereof 上海医药工业研究院 2021-07-02 CN disclosed
CN-110467638-A A kind of double amino Chloropyrimide class compounds containing m-chloroaniline class substituent group, preparation method and applications BEIJING SAITE MINGQIANG MEDICINE TECH CO LTD 2019-11-19 CN disclosed
WO-2012115479-A2 DIAMINOPYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 2012-08-30 WO disclosed
EP-1981856-A2 PYRIMIDINE DERIVATIVES AstraZeneca AB (SE) 2008-10-22 EP disclosed
WO-2007085833-A2 PYRIMIDINE DERIVATIVES ASTRAZENECA AB (SE) 2007-08-02 WO disclosed
EP-0674627-A1 PYRIMIDINE, PYRIDINE, PTERIDINONE AND INDAZOLE DERIVATIVES AS ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-10-04 EP disclosed
WO-1994014780-A1 PYRIMIDINE, PYRIDINE, PTERIDINONE AND INDAZOLE DERIVATIVES AS ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1994-07-07 WO disclosed