SCHEMBL29664332

SCHEMBL29664332

Nc1cccc(-c2cnn(-c3ccccc3)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.53
TSHR P16473 1/20 0.47
MEN1 O00255 3/20 0.46
KMT2A Q03164 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
MAP4K4 O95819 2/20 0.46
GAA P10253 1/20 0.46
GRM4 Q14833 7/20 0.46
PSIP1 O75475 1/20 0.45
AXL P30530 1/20 0.45
MKNK1 Q9BUB5 1/20 0.45
MKNK2 Q9HBH9 1/20 0.45
HSP90AA1 P07900 1/20 0.45
HTR2B P41595 1/20 0.44
MTNR1A P48039 1/20 0.44
KCNH2 Q12809 1/20 0.44
GRM2 Q14416 1/20 0.44
MECP2 P51608 1/20 0.42
HPGDS O60760 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23144535 1.00 MAOA (0.53) MAOATSHRMEN1KMT2ANPC1
SCHEMBL23144559 0.94 MAOA (0.55) MAOATSHRMEN1KMT2ANPC1
SCHEMBL29664328 0.88 MKNK1 (0.50) MAOAMEN1KMT2ANPC1RAB9A
SCHEMBL23144521 0.88 MKNK1 (0.50) MAOAMEN1KMT2ANPC1RAB9A
SCHEMBL23144544 0.86 GRM4 (0.47) MAOAMEN1KMT2ANPC1RAB9A
SCHEMBL29664194 0.86 MAP4K4 (0.44) MAOAMEN1KMT2ANPC1RAB9A
SCHEMBL23144576 0.86 MAP4K4 (0.44) MAOAMEN1KMT2ANPC1RAB9A
SCHEMBL29664364 0.86 GRM4 (0.47) MAOAMEN1KMT2ANPC1RAB9A
SCHEMBL23144557 0.83 NTRK1 (0.57) MAOATSHRMEN1KMT2ANPC1
SCHEMBL23144571 0.83 MAPKAPK2 (0.56) TSHRMEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114728909-A Composition for preventing or treating cancer comprising novel trifluoromethylphenylpyrazole derivative as active ingredient 韩国原子力医学院 2022-07-08 CN disclosed
EP-4015506-A2 COMPOSITION FOR PREVENTING OR TREATING CANCER, CONTAINING NOVEL TRIFLUOROMETHYL PHENYL PYRAZOLE DERIVATIVE AS ACTIVE INGREDIENT Korea Institute of Radiological & Medical Sciences (KR) 2022-06-22 EP disclosed