SCHEMBL29664740

SCHEMBL29664740

N#Cc1ccc(CN(CCN)Cc2ccc(C#N)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 2/20 0.55
CYP2A6 P11509 1/20 0.45
RORC P51449 1/20 0.44
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
IDO1 P14902 2/20 0.41
NSD2 O96028 2/20 0.39
HRH3 Q9Y5N1 2/20 0.38
MEP1B Q16820 1/20 0.38
CYP19A1 P11511 3/20 0.38
KCNJ1 P48048 1/20 0.38
KCNH2 Q12809 1/20 0.38
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4410040 0.96 LOXL2 (0.55) LOXL2CYP2A6RORCCRHBPCRHR2
SCHEMBL29278097 0.90 LOXL2 (0.48) LOXL2CYP2A6RORCNSD2HRH3
SCHEMBL15831721 0.82 HRH3 (0.59) LOXL2CYP2A6RORCCRHBPCRHR2
SCHEMBL4406268 0.79 HRH3 (0.50) HRH3
SCHEMBL6263851 0.78 LOXL2 (0.47) LOXL2CYP2A6RORCCRHBPCRHR2
SCHEMBL19088665 0.78 HRH3 (0.64) LOXL2CYP2A6RORCNSD2HRH3
SCHEMBL6263660 0.77 LOXL2 (0.45) LOXL2CYP2A6RORCCRHBPCRHR2
SCHEMBL2201240 0.77 RORC (0.53) CYP2A6RORCHRH3
SCHEMBL541669 0.76 HRH3 (0.59) LOXL2CYP2A6RORCHRH3
SCHEMBL27909746 0.74 CYP1A2 (0.52) CYP2A6RORCIDO1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114507175-A Novel inhibitors of hypnotic proteins alpha and beta 维沃里翁治疗股份有限公司 2022-05-17 CN disclosed