SCHEMBL29673145

SCHEMBL29673145

O=C1CCCc2c(OC(F)(F)F)cccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.47
ADRB1 P08588 1/20 0.47
HTR1A P08908 1/20 0.47
ADRB3 P13945 1/20 0.47
TSHR P16473 1/20 0.47
SLC6A4 P31645 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
MRGPRX4 Q96LA9 1/20 0.47
CYP2A6 P11509 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
HPGD P15428 1/20 0.40
ABCB1 P08183 2/20 0.39
BRD4 O60885 2/20 0.38
BRAF P15056 1/20 0.38
GPR174 Q9BXC1 1/20 0.36
POLB P06746 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SCN9A Q15858 1/20 0.36
ANO1 Q5XXA6 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24543427 1.00 ADRB2 (0.47) ADRB2ADRB1HTR1AADRB3TSHR
SCHEMBL1508672 0.90 ABCB1 (0.43) ADRB2ADRB1HTR1AADRB3TSHR
SCHEMBL15319609 0.80 MRGPRX4 (0.53) ADRB2ADRB1HTR1AADRB3TSHR
SCHEMBL2729107 0.79 MRGPRX4 (0.46) ADRB2ADRB1HTR1AADRB3TSHR
SCHEMBL8827446 0.79 ADRB2 (0.42) ADRB2ADRB1HTR1AADRB3TSHR
SCHEMBL264705 0.78 BRD4 (0.54) ADRB2ADRB1HTR1AADRB3TSHR
SCHEMBL29802310 0.78 BRD4 (0.54) ADRB2ADRB1HTR1AADRB3TSHR
SCHEMBL5692114 0.76 RXRB (0.42) MRGPRX4ANO1
SCHEMBL9489544 0.75 MRGPRX4 (0.45) ADRB2ADRB1HTR1AADRB3TSHR
SCHEMBL1508383 0.75 CYP2A6 (0.44) ADRB2ADRB1HTR1AADRB3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022127827-A1 KRASG12C PROTEIN MUTATION INHIBITOR AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 上海维申医药有限公司 2022-06-23 WO disclosed
CN-114644631-A KRAS G12C protein mutation inhibitor, preparation method thereof, pharmaceutical composition and application thereof 上海维申医药有限公司 2022-06-21 CN disclosed