SCHEMBL29673151

SCHEMBL29673151

O=C1CCCc2c(Cl)cc(F)cc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.42
MAOA P21397 4/20 0.37
MAOB P27338 4/20 0.37
PRKCI P41743 1/20 0.37
MAPT P10636 4/20 0.34
MAPK1 P28482 3/20 0.34
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 3/20 0.34
HSD17B10 Q99714 3/20 0.34
GAA P10253 2/20 0.34
ALOX15 P16050 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
LMNA P02545 2/20 0.34
POLB P06746 1/20 0.34
BRD4 O60885 3/20 0.34
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CYP2A6 P11509 1/20 0.33
PARP1 P09874 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24543321 1.00 NOTUM (0.42) NOTUMMAOAMAOBPRKCIMAPT
SCHEMBL29673147 0.89 NOTUM (0.48) NOTUMMAOAMAOBMAPTKDM4E
SCHEMBL2262470 0.89 NOTUM (0.48) NOTUMMAOAMAOBMAPTKDM4E
SCHEMBL8459403 0.81 MAOA (0.44) MAOAMAOBPRKCIMAPK1KDM4E
SCHEMBL7815325 0.81 MEN1 (0.49) NOTUMMAOAMAOBPRKCIMAPT
SCHEMBL30070487 0.81 MAOA (0.44) MAOAMAOBPRKCIMAPK1KDM4E
SCHEMBL11460490 0.79 BRD4 (0.38) MAOAMAOBPRKCIMAPTMAPK1
SCHEMBL30917672 0.78 MAOA (0.41) MAOAMAOBPRKCIMAPTMAPK1
SCHEMBL29673079 0.78 NOTUM (0.42) NOTUMMAOAMAOBPRKCIMAPT
SCHEMBL11741693 0.78 NOTUM (0.42) NOTUMMAOAMAOBPRKCIMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022127827-A1 KRASG12C PROTEIN MUTATION INHIBITOR AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 上海维申医药有限公司 2022-06-23 WO disclosed
CN-114644631-A KRAS G12C protein mutation inhibitor, preparation method thereof, pharmaceutical composition and application thereof 上海维申医药有限公司 2022-06-21 CN disclosed