SCHEMBL29680469

SCHEMBL29680469

COC(=O)C(N)CCCCNCc1ccc(-c2nc(-c3ccc(CNCCCCC(N)C(=O)OC)cc3)c3ccn(C)c3n2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP8 Q6V1X1 1/20 0.38
DPP9 Q86TI2 1/20 0.38
DPP7 Q9UHL4 1/20 0.38
HRH4 Q9H3N8 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
S1PR2 O95136 2/20 0.34
S1PR1 P21453 2/20 0.34
S1PR3 Q99500 2/20 0.34
LPAR2 Q9HBW0 2/20 0.34
TPH1 P17752 2/20 0.34
CYP3A4 P08684 1/20 0.33
MAPT P10636 1/20 0.33
TLR7 Q9NYK1 3/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
MMP1 P03956 1/20 0.33
CYP2D6 P10635 1/20 0.33
MMP9 P14780 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL29680414 0.97 DPP7 (0.38) DPP8DPP9DPP7HRH4HRH3
Oxalic Acid SCHEMBL29680599 0.77 TERT (0.40) S1PR2S1PR1S1PR3LPAR2TSHR
SCHEMBL29680699 0.76 LMNA (0.43) HRH4HRH3S1PR2S1PR1S1PR3
Oxalic Acid SCHEMBL29680295 0.75 AKT1 (0.46) S1PR2S1PR1S1PR3LPAR2CYP3A4
SCHEMBL29680354 0.73 AKT1 (0.48) HRH4HRH3S1PR2S1PR1S1PR3
Hydrochloric Acid SCHEMBL8527393 0.68 DPP8 (0.54) DPP8DPP9DPP7MAPT
Oxalic Acid SCHEMBL29680335 0.67 TERT (0.38) S1PR2S1PR1S1PR3LPAR2TSHR
SCHEMBL24528705 0.67 CYP2A6 (0.39) CYP3A4MAPT
SCHEMBL29681096 0.67 CYP2A6 (0.39) CYP3A4MAPT
Oxalic Acid SCHEMBL29680355 0.66 KDM4E (0.41) CYP3A4CYP2D6TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4263539-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2023-10-25 EP claimed
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO claimed
EP-4263539-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2023-10-25 EP disclosed
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed