SCHEMBL29680684

SCHEMBL29680684

CN1CCN(CCCCNCc2ccc(-c3cc(-c4ccc(CNCCCCN5CCN(C)CC5)cc4)c4cc[nH]c4n3)cc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.48
AKT2 P31751 1/20 0.48
JAK1 P23458 7/20 0.44
IKBKB O14920 2/20 0.40
CHUK O15111 2/20 0.40
ABL1 P00519 2/20 0.40
INSR P06213 2/20 0.40
CDK2 P24941 2/20 0.40
FLT3 P36888 2/20 0.40
MAP3K11 Q16584 2/20 0.40
TNIK Q9UKE5 4/20 0.37
SGK1 O00141 1/20 0.37
AURKA O14965 1/20 0.37
PRKAB2 O43741 1/20 0.37
ROCK2 O75116 1/20 0.37
NTRK1 P04629 1/20 0.37
LCK P06239 1/20 0.37
CDK1 P06493 1/20 0.37
IGF1R P08069 1/20 0.37
MET P08581 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL29680336 0.94 AKT1 (0.46) AKT1AKT2JAK1
SCHEMBL29680686 0.80 TERT (0.41) JAK1IKBKBCHUKCDK2
SCHEMBL29681210 0.78 JAK1 (0.39) JAK1IKBKBCHUKABL1INSR
SCHEMBL24528644 0.78 JAK1 (0.39) JAK1IKBKBCHUKABL1INSR
SCHEMBL29680455 0.78 AKT1 (0.48) AKT1AKT2IKBKBCHUKABL1
Oxalic Acid SCHEMBL29680687 0.75 JAK1 (0.43) JAK1IKBKBCHUKCDK2
Oxalic Acid SCHEMBL29680236 0.74 AKT1 (0.46) AKT1AKT2JAK1AURKAAURKB
SCHEMBL3181062 0.72 CYP2C19 (0.55) AKT1AKT2CYP3A4
SCHEMBL3171946 0.69 DPP7 (0.57) AKT1AKT2CYP3A4
SCHEMBL4418818 0.68 CHRM2 (0.51) AKT1AKT2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4263539-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2023-10-25 EP claimed
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO claimed
EP-4263539-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2023-10-25 EP disclosed
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed