SCHEMBL24528644

SCHEMBL24528644

CN1CCN(CCCC/N=C\c2ccc(-c3cc(-c4ccc(/C=N/CCCCN5CCN(C)CC5)cc4)nc4[nH]ccc34)cc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 7/20 0.39
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
IKBKB O14920 2/20 0.35
CHUK O15111 2/20 0.35
ABL1 P00519 2/20 0.35
INSR P06213 2/20 0.35
CDK2 P24941 2/20 0.35
FLT3 P36888 2/20 0.35
MAP3K11 Q16584 2/20 0.35
ALOX15 P16050 1/20 0.33
PRKCQ Q04759 1/20 0.33
PRKCD Q05655 1/20 0.33
TNIK Q9UKE5 3/20 0.33
RPS6KA3 P51812 3/20 0.33
SGK1 O00141 1/20 0.33
AURKA O14965 1/20 0.33
PRKAB2 O43741 1/20 0.33
ROCK2 O75116 1/20 0.33
NTRK1 P04629 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29681210 1.00 JAK1 (0.39) JAK1KDM4EALDH1A1IKBKBCHUK
SCHEMBL24528665 0.81 NEK1 (0.36) JAK1ALDH1A1IKBKBCHUKSYK
SCHEMBL29680982 0.81 NEK1 (0.36) JAK1ALDH1A1IKBKBCHUKSYK
SCHEMBL29680615 0.79 KDM4E (0.39) KDM4EALDH1A1IKBKBCHUKABL1
SCHEMBL24528663 0.79 KDM4E (0.39) KDM4EALDH1A1IKBKBCHUKABL1
SCHEMBL29680684 0.78 AKT1 (0.48) JAK1IKBKBCHUKABL1INSR
Oxalic Acid SCHEMBL29680336 0.74 AKT1 (0.46) JAK1KDM4EALDH1A1
SCHEMBL24528632 0.68 CYP2A6 (0.39) JAK1ALDH1A1IKBKBCHUKPRKCQ
SCHEMBL29680885 0.68 CYP2A6 (0.39) JAK1ALDH1A1IKBKBCHUKPRKCQ
SCHEMBL24528660 0.65 KDM4E (0.40) KDM4EALDH1A1ALOX15MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed