SCHEMBL29680773

SCHEMBL29680773

CN1CCN(CCCN=Cc2ccc(-c3nc(Cl)nc4c3ccn4-c3ccccc3)cc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 4/20 0.36
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
MAPT P10636 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MAPK1 P28482 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
USP2 O75604 2/20 0.33
CASP1 P29466 2/20 0.33
CASP7 P55210 2/20 0.33
SLC2A1 P11166 1/20 0.33
LMNA P02545 1/20 0.32
MAP4K1 Q92918 1/20 0.32
FLT3 P36888 1/20 0.31
BCL2L1 Q07817 1/20 0.31
SIGMAR1 Q99720 3/20 0.31
RAD52 P43351 1/20 0.31
TP53 P04637 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24528659 1.00 ALDH1A1 (0.36) ALDH1A1KDM4ENPC1RAB9AMAPT
SCHEMBL24528667 0.96 ALDH1A1 (0.36) ALDH1A1KDM4ENPC1RAB9AMAPT
SCHEMBL29681267 0.96 ALDH1A1 (0.36) ALDH1A1KDM4ENPC1RAB9AMAPT
SCHEMBL29680554 0.90 RAD52 (0.37) ALDH1A1KDM4ENPC1RAB9AMAPT
SCHEMBL24528648 0.90 RAD52 (0.37) ALDH1A1KDM4ENPC1RAB9AMAPT
SCHEMBL24528661 0.88 RAD52 (0.36) ALDH1A1KDM4ENPC1RAB9AMAPT
SCHEMBL24528671 0.87 DRD2 (0.36) ALDH1A1KDM4ENPC1RAB9AMAPT
SCHEMBL24528649 0.86 RAD52 (0.34) ALDH1A1KDM4ENPC1RAB9AMAPT
SCHEMBL24528583 0.84 KDM4E (0.38) ALDH1A1KDM4ELMNA
SCHEMBL29680660 0.84 KDM4E (0.38) ALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4263539-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2023-10-25 EP disclosed
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed