SCHEMBL29683161

SCHEMBL29683161

FC(F)(F)Cc1cc(Br)ccn1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
SLC22A12 Q96S37 1/20 0.33
RAD51 Q06609 1/20 0.32
LOXL2 Q9Y4K0 2/20 0.32
HRH4 Q9H3N8 1/20 0.31
LOX P28300 1/20 0.31
SYK P43405 1/20 0.31
NOS3 P29474 1/20 0.31
NOS2 P35228 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
MAPT P10636 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23617121 1.00 KDM4E (0.37) KDM4EALDH1A1SMN1; SMN2SLC22A12RAD51
SCHEMBL19783105 0.77 KDM4E (0.43) KDM4EALDH1A1SMN1; SMN2CYP1A2CYP3A4
SCHEMBL31278153 0.77
SCHEMBL23235054 0.77
SCHEMBL20197189 0.76 HDAC8 (0.36) LOXL2LOXNOS3NOS2
SCHEMBL16548463 0.76 UHRF1 (0.45) KDM4EALDH1A1SMN1; SMN2SYKNOS3
SCHEMBL25203651 0.74 LOXL2 (0.59) LOXL2LOXSYK
SCHEMBL26192789 0.74 NOS3 (0.50) KDM4ELOXL2LOXNOS3NOS2
SCHEMBL31706588 0.74 SIRT2 (0.38) KDM4EALDH1A1
SCHEMBL29898951 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022127756-A1 COMPOUNDS AS CASEIN KINASE INHIBITORS Gritscience Biopharmaceuticals Co., Ltd. (CN) 2022-06-23 WO disclosed