Levomepromazine

Levomepromazine

SCHEMBL29697036

COc1ccc2c(c1)N(C[C@H](C)CN(C)C)c1ccccc1S2.O=C(O)/C=C\C(=O)O

nearest known ligand 0.82

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2DRD3DRD4

The experimentally established mechanism targets of Levomepromazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 known ✓ P35462 4/20 0.82
DRD2 known ✓ P14416 2/20 0.46
DRD4 known ✓ P21917 1/20 0.43
LMNA P02545 5/20 0.82
CHRM2 P08172 4/20 0.82
HTR1A P08908 4/20 0.82
CHRM1 P11229 4/20 0.82
ADRA1A P35348 4/20 0.82
OPRM1 P35372 4/20 0.82
KCNH2 Q12809 4/20 0.82
CYP2D6 P10635 4/20 0.82
ADRA2A P08913 3/20 0.82
DRD1 P21728 3/20 0.82
CYP3A4 P08684 3/20 0.82
MAPK1 P28482 3/20 0.82
TBXA2R P21731 2/20 0.82
CYP1A2 P05177 2/20 0.82
PTGS1 P23219 2/20 0.82
GFER P55789 1/20 0.62
SLC6A2 P23975 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Levomepromazine SCHEMBL29727144 1.00 LMNA (0.82) LMNACHRM2HTR1ACHRM1ADRA1A
Levomepromazine SCHEMBL218717 1.00 LMNA (0.82) LMNACHRM2HTR1ACHRM1ADRA1A
Levomepromazine SCHEMBL27701483 0.93 LMNA (0.88) LMNACHRM2HTR1ACHRM1ADRA1A
Levomepromazine SCHEMBL29508092 0.91 CYP2D6 (1.00) LMNACHRM2HTR1ACHRM1ADRA1A
Levomepromazine SCHEMBL8762418 0.91 CYP2D6 (1.00) LMNACHRM2HTR1ACHRM1ADRA1A
Dextromepromazine SCHEMBL23859840 0.91 CYP2D6 (1.00) LMNACHRM2HTR1ACHRM1ADRA1A
Levomepromazine SCHEMBL6944555 0.91 CYP2D6 (1.00) LMNACHRM2HTR1ACHRM1ADRA1A
Levomepromazine SCHEMBL29425180 0.91 CYP2D6 (1.00) LMNACHRM2HTR1ACHRM1ADRA1A
Levomepromazine SCHEMBL25462 0.91 CYP2D6 (1.00) LMNACHRM2HTR1ACHRM1ADRA1A
Levomepromazine SCHEMBL29384983 0.91 CYP2D6 (1.00) LMNACHRM2HTR1ACHRM1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12410474-B2 Methods, kits, and devices for diagnosing, prognosing, and treating psychiatric disorders in a patient NORTHWESTERN UNIVERSITY (US) 2025-09-09 US disclosed
WO-2025033273-A1 DISPENSATION CONTROL DEVICE, MEDICINE DISPENSATION SYSTEM, AND MEDICINE DISPENSATION PROGRAM 株式会社湯山製作所 2025-02-13 WO disclosed
US-20240285549-A1 CANNABIS OIL COMPOSITIONS AND METHODS FOR PREPARATION THEREOF CONSTANCE THERAPEUTICS, INC. (US) 2024-08-29 US disclosed
US-20240033312-A1 CANNABIS OIL EXTRACTS AND COMPOSITIONS CONSTANCE THERAPEUTICS, INC. (US) 2024-02-01 US disclosed
US-20230386637-A1 Polymorphisms for Predicting Treatment Response to Antipsychotic Drugs and Identifying New Drug Targets NORTHWESTERN UNIVERSITY 2023-11-30 US disclosed
US-11596618-B2 Oral cannabinoid delivery formulations with mouthfeel experience enhancers Resurgent Biosciences, Inc. (US) 2023-03-07 US disclosed
US-20220331344-A1 ORAL FORMULATIONS OF PSYCHOTROPIC MACROFUNGUS BOTANICAL EXTRACTS WITH MOUTHFEEL EXPERIENCE ENHANCERS CHICAGO ATLANTIC ADMIN, LLC 2022-10-20 US disclosed
US-20220177970-A1 METHODS, KITS, AND DEVICES FOR DIAGNOSING, PROGNOSING, AND TREATING PSYCHIATRIC DISORDERS IN A PATIENT NORTHWESTERN UNIVERSITY 2022-06-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240033312-A1 CANNABIS OIL EXTRACTS AND COMPOSITIONS CNR2, CNR1, DNER DRD3 332/4885DRD2 213/4885DRD4 229/4885
US-20240285549-A1 CANNABIS OIL COMPOSITIONS AND METHODS FOR PREPARATION THEREOF CNR1, CNR2, PROC DRD3 311/4885DRD2 215/4885DRD4 248/4885
US-20220331344-A1 ORAL FORMULATIONS OF PSYCHOTROPIC MACROFUNGUS BOTANICAL EXTRACTS WITH MOUTHFEEL EXPERIENCE ENHANCERS MB, MLEC, NISCH DRD3 583/4885DRD2 145/4885DRD4 521/4885
US-11596618-B2 Oral cannabinoid delivery formulations with mouthfeel experience enhancers CNR2, CNR1, CPNE4 DRD3 400/4885DRD2 224/4885DRD4 382/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.