SCHEMBL29698205

SCHEMBL29698205

COc1cc(C)cnc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.43
ALDH1A1 P00352 4/20 0.41
CCR1 P32246 1/20 0.35
CCR5 P51681 1/20 0.35
CCR8 P51685 1/20 0.35
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
PDGFRB P09619 6/20 0.35
PDGFRA P16234 6/20 0.35
CYP3A4 P08684 1/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
ALOX12 P18054 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4373862 1.00 ACHE (0.43) ACHEALDH1A1CCR1CCR5CCR8
SCHEMBL21446936 0.80 ALDH1A1 (0.43) ALDH1A1PDGFRBPDGFRACYP3A4CYP2C9
SCHEMBL10084731 0.80 ACHE (0.44) ACHEALDH1A1CCR1CCR5CCR8
SCHEMBL24476817 0.78 ALDH1A1 (0.41) ALDH1A1CCR1CCR5CCR8PDGFRB
SCHEMBL10084727 0.77 ACHE (0.46) ACHEALDH1A1CCR1CCR5CCR8
SCHEMBL29483025 0.77 ALDH1A1 (0.40) ALDH1A1MEN1POLBMAPTALOX12
SCHEMBL2118826 0.77 ALDH1A1 (0.40) ALDH1A1MEN1POLBMAPTALOX12
SCHEMBL117167 0.77 ALDH1A1 (0.40) ALDH1A1PDGFRBPDGFRAMEN1MAPT
SCHEMBL19555271 0.77 CYP3A4 (0.45) ALDH1A1PDGFRBPDGFRACYP3A4MAPT
SCHEMBL10112981 0.74 ACHE (0.43) ACHEALDH1A1CCR1CCR5CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4010334-A1 HETEROCYCLIC WDR5 INHIBITORS AS ANTI-CANCER COMPOUNDS Novartis AG (CH) 2022-06-15 EP disclosed