SCHEMBL29699319

SCHEMBL29699319

Nc1nc(C(F)(F)F)c(-c2ccco2)nc1C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 2/20 0.50
PLAU P00749 2/20 0.50
MAPT P10636 6/20 0.42
KMT2A Q03164 6/20 0.42
MEN1 O00255 5/20 0.42
POLB P06746 5/20 0.42
ALDH1A1 P00352 5/20 0.42
L3MBTL1 Q9Y468 4/20 0.42
THRB P10828 2/20 0.42
NSD2 O96028 1/20 0.42
GAA P10253 1/20 0.42
PABPC1 P11940 1/20 0.42
TNNI3 P19429 1/20 0.42
TNNT2 P45379 1/20 0.42
TNNC1 P63316 1/20 0.42
ADORA2A P29274 3/20 0.41
KDM4E B2RXH2 4/20 0.40
BLM P54132 3/20 0.40
HPGD P15428 3/20 0.40
TDP1 Q9NUW8 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2371359 1.00 CFTR (0.50) CFTRPLAUMAPTKMT2AMEN1
SCHEMBL14631665 0.84 CFTR (0.47) CFTRPLAUMAPTKMT2AMEN1
SCHEMBL29699257 0.74 CACNA1B (0.54) CFTRMAPTKMT2AMEN1POLB
SCHEMBL2372725 0.74 CACNA1B (0.54) CFTRMAPTKMT2AMEN1POLB
SCHEMBL2371668 0.73 PLAU (0.36) CFTRPLAUMAPTALDH1A1KDM4E
SCHEMBL2371983 0.71 MAPT (0.46) CFTRMAPTKMT2AMEN1POLB
SCHEMBL22573733 0.71 POLB (0.50) PLAUMAPTKMT2AMEN1POLB
SCHEMBL4584998 0.70 ADORA2A (0.57) PLAUMAPTKMT2AMEN1POLB
SCHEMBL10374405 0.69 ALDH1A1 (0.52) CFTRPLAUMAPTKMT2AMEN1
SCHEMBL4584246 0.68 ADORA2A (0.44) PLAUMAPTKMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3980121-A1 PYRIDINE AND PYRAZINE DERIVATIVE FOR THE TREATMENT OF CF, COPD, AND BRONCHIECTASIS Novartis AG (CH) 2022-04-13 EP disclosed