SCHEMBL29699381

SCHEMBL29699381

COC(=O)c1nc(Br)c(C(F)(F)F)cc1-n1c(C)ccc1C

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CFTR P13569 10/20 0.45
NOTUM Q6P988 2/20 0.43
MYC P01106 2/20 0.42
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
RBP4 P02753 2/20 0.39
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2372633 1.00 CFTR (0.45) CFTRNOTUMMYCALDH1A1KDM4E
SCHEMBL13518970 0.95 CFTR (0.42) CFTRNOTUMMYCALDH1A1KDM4E
SCHEMBL2383885 0.86 MYC (0.43) CFTRNOTUMMYCALDH1A1KDM4E
SCHEMBL2372372 0.86 MYC (0.43) CFTRNOTUMMYCALDH1A1KDM4E
SCHEMBL29699241 0.86 CFTR (0.45) CFTRMYCHSD17B10
SCHEMBL2372056 0.86 CFTR (0.45) CFTRMYCHSD17B10
SCHEMBL2381481 0.85 CFTR (0.42) CFTRNOTUMMYCALDH1A1KDM4E
SCHEMBL12295762 0.85 CFTR (0.40) CFTRNOTUMMYCALDH1A1KDM4E
SCHEMBL2372480 0.81 CFTR (0.40) CFTRNOTUMMYCALDH1A1KDM4E
SCHEMBL2372871 0.81 CFTR (0.45) CFTRNOTUMMYCALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3980121-A1 PYRIDINE AND PYRAZINE DERIVATIVE FOR THE TREATMENT OF CF, COPD, AND BRONCHIECTASIS Novartis AG (CH) 2022-04-13 EP disclosed