SCHEMBL29699241

SCHEMBL29699241

Cc1ccc(C)n1-c1cc(C(F)(F)F)c(Br)nc1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CFTR P13569 7/20 0.45
MYC P01106 12/20 0.43
NR4A1 P22736 3/20 0.43
ESR1 P03372 1/20 0.39
ALOX15 P16050 1/20 0.39
PTPN7 P35236 1/20 0.39
HSD17B10 Q99714 1/20 0.39
GRIA1 P42261 1/20 0.38
GRIA2 P42262 1/20 0.38
GRIA3 P42263 1/20 0.38
GRIA4 P48058 1/20 0.38
PTPN1 P18031 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2372056 1.00 CFTR (0.45) CFTRMYCNR4A1ESR1ALOX15
SCHEMBL13518970 0.92 CFTR (0.42) CFTRMYCNR4A1HSD17B10
SCHEMBL2372633 0.86 CFTR (0.45) CFTRMYCHSD17B10
SCHEMBL29699381 0.86 CFTR (0.45) CFTRMYCHSD17B10
SCHEMBL2372656 0.85 MYC (0.44) CFTRMYCNR4A1ESR1ALOX15
SCHEMBL29699221 0.85 MYC (0.44) CFTRMYCNR4A1ESR1ALOX15
SCHEMBL2373031 0.82 MYC (0.44) CFTRMYCNR4A1ESR1ALOX15
SCHEMBL12295762 0.81 CFTR (0.40) CFTRMYCNR4A1GRIA1GRIA2
SCHEMBL28800852 0.81 AGBL2 (0.43) CFTRMYCNR4A1ESR1ALOX15
SCHEMBL2372906 0.79 CFTR (0.44) CFTRMYCESR1ALOX15PTPN7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3980121-A1 PYRIDINE AND PYRAZINE DERIVATIVE FOR THE TREATMENT OF CF, COPD, AND BRONCHIECTASIS Novartis AG (CH) 2022-04-13 EP disclosed