SCHEMBL29699759

SCHEMBL29699759

Cc1ccc(NC(=O)c2cc(C)n(Cc3cccc(Br)c3)n2)cc1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.79
KMT2A Q03164 2/20 0.79
AURKA O14965 1/20 0.54
RPS6KB1 P23443 1/20 0.54
POLB P06746 1/20 0.53
NPSR1 Q6W5P4 3/20 0.52
P2RY14 Q15391 3/20 0.50
CYP3A4 P08684 3/20 0.50
CYP2C9 P11712 3/20 0.50
LMNA P02545 3/20 0.50
PTGER1 P34995 4/20 0.49
MAPT P10636 2/20 0.48
MAPK1 P28482 1/20 0.47
HTR1E P28566 1/20 0.47
S1PR3 Q99500 1/20 0.47
CYP2C19 P33261 1/20 0.46
STAT3 P40763 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KDM4E B2RXH2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29700093 0.92 MEN1 (0.67) MEN1KMT2AAURKARPS6KB1POLB
SCHEMBL29699847 0.91 MEN1 (0.66) MEN1KMT2AAURKARPS6KB1POLB
SCHEMBL29699779 0.89 MEN1 (0.64) MEN1KMT2AAURKARPS6KB1POLB
SCHEMBL29699739 0.89 CYP3A4 (0.64) MEN1KMT2AAURKARPS6KB1POLB
SCHEMBL1899756 0.89 MEN1 (1.00) MEN1KMT2AAURKARPS6KB1POLB
SCHEMBL29699842 0.86 CYP3A4 (0.65) MEN1KMT2AAURKARPS6KB1POLB
SCHEMBL29699837 0.85 MEN1 (0.58) MEN1KMT2AAURKARPS6KB1POLB
SCHEMBL1902344 0.83 MEN1 (0.78) MEN1KMT2AAURKARPS6KB1NPSR1
SCHEMBL1897273 0.82 MEN1 (0.80) MEN1KMT2AAURKARPS6KB1NPSR1
4-Bromoaniline SCHEMBL7739202 0.81 MEN1 (0.80) MEN1KMT2AAURKARPS6KB1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114685371-A Pyrazole carboxamide derivatives, their preparation and use 四川大学 2022-07-01 CN disclosed