SCHEMBL29699847

SCHEMBL29699847

Cc1cc(C(=O)Nc2ccc(F)cc2)nn1Cc1cccc(Br)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.66
KMT2A Q03164 1/20 0.66
PTGER1 P34995 5/20 0.58
MAPK1 P28482 2/20 0.52
NPSR1 Q6W5P4 2/20 0.52
HTR1E P28566 1/20 0.52
S1PR3 Q99500 1/20 0.52
AURKA O14965 1/20 0.52
RPS6KB1 P23443 1/20 0.52
CYP3A4 P08684 3/20 0.51
CYP2C9 P11712 3/20 0.51
NPY5R Q15761 2/20 0.50
LMNA P02545 2/20 0.48
POLB P06746 1/20 0.48
MAPT P10636 2/20 0.48
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29699759 0.91 MEN1 (0.79) MEN1KMT2APTGER1MAPK1NPSR1
SCHEMBL29700093 0.90 MEN1 (0.67) MEN1KMT2APTGER1AURKARPS6KB1
SCHEMBL29699739 0.89 CYP3A4 (0.64) MEN1KMT2APTGER1AURKARPS6KB1
SCHEMBL29699779 0.88 MEN1 (0.64) MEN1KMT2APTGER1AURKARPS6KB1
SCHEMBL29699842 0.86 CYP3A4 (0.65) MEN1KMT2APTGER1AURKARPS6KB1
SCHEMBL29699837 0.83 MEN1 (0.58) MEN1KMT2APTGER1AURKARPS6KB1
SCHEMBL1899756 0.80 MEN1 (1.00) MEN1KMT2APTGER1NPSR1AURKA
SCHEMBL29699803 0.79 PTGER1 (0.69) MEN1KMT2APTGER1P2RY14
SCHEMBL29699784 0.75 CYP19A1 (0.57) MEN1KMT2APTGER1LMNAPOLB
SCHEMBL29699827 0.75 MEN1 (0.73) MEN1KMT2APTGER1AURKARPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114685371-A Pyrazole carboxamide derivatives, their preparation and use 四川大学 2022-07-01 CN disclosed