SCHEMBL29721920

SCHEMBL29721920

Cc1cccc(-c2ncc(O)c(Nc3ccncc3)n2)n1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 17/20 0.59
MAPK14 Q16539 1/20 0.59
TGFBR2 P37173 3/20 0.56
BUB1 O43683 3/20 0.44
CYP3A4 P08684 1/20 0.43
CYP2C8 P10632 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28734419 1.00 TGFBR1 (0.59) TGFBR1MAPK14TGFBR2BUB1CYP3A4
SCHEMBL28734420 0.82 TGFBR1 (0.57) TGFBR1MAPK14TGFBR2BUB1
SCHEMBL6684058 0.74 TGFBR1 (1.00) TGFBR1MAPK14CYP3A4
SCHEMBL13727304 0.74 CCR1 (0.50) TGFBR1MAPK14
SCHEMBL14726013 0.72 TGFBR1 (0.76) TGFBR1MAPK14TGFBR2
SCHEMBL18414358 0.72 TGFBR1 (1.00) TGFBR1TGFBR2
SCHEMBL18397543 0.69 TGFBR1 (0.83) TGFBR1MAPK14TGFBR2
SCHEMBL20434739 0.69 TGFBR1 (0.83) TGFBR1MAPK14TGFBR2
SCHEMBL14731231 0.69 TGFBR1 (0.70) TGFBR1MAPK14TGFBR2CYP3A4
SCHEMBL18414916 0.68 TGFBR1 (1.00) TGFBR1MAPK14TGFBR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114380845-A Heterocyclic-fused compound, pharmaceutical composition containing same, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2022-04-22 CN disclosed