SCHEMBL29723979

SCHEMBL29723979

Nc1nc2ccc(-c3ccc4ncncc4c3)cc2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.53
PIK3CA P42336 2/20 0.52
PIK3CD O00329 1/20 0.52
TDO2 P48775 1/20 0.48
PLAU P00749 1/20 0.47
HTR3E A5X5Y0 1/20 0.47
HTR3B O95264 1/20 0.47
HTR3A P46098 1/20 0.47
BACE1 P56817 1/20 0.47
HTR3D Q70Z44 1/20 0.47
HTR3C Q8WXA8 1/20 0.47
FGFR4 P22455 1/20 0.43
ALDH1A1 P00352 3/20 0.42
TDP1 Q9NUW8 2/20 0.42
MTOR P42345 1/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
MASP2 O00187 1/20 0.41
NUDT1 P36639 1/20 0.41
AOC3 Q16853 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8644295 0.80 PIK3CA (0.73) EGFRPIK3CAPIK3CDTDO2FGFR4
SCHEMBL29723993 0.76 EGFR (0.61) EGFRPIK3CAPIK3CDTDO2FGFR4
SCHEMBL11712219 0.74 ALDH1A1 (0.58) PIK3CAPLAUHTR3EHTR3BHTR3A
SCHEMBL28178788 0.74 EGFR (0.67) EGFRPIK3CAPIK3CDTDO2FGFR4
SCHEMBL3042419 0.73 PIK3CD (0.63) EGFRPIK3CAPIK3CDTDO2FGFR4
SCHEMBL20687402 0.73 PIK3CD (0.73) EGFRPIK3CAPIK3CDTDO2BACE1
SCHEMBL30669824 0.72 PIK3CA (0.62) EGFRPIK3CAPIK3CDTDO2ALDH1A1
SCHEMBL27892456 0.72 PIK3CA (0.62) EGFRPIK3CAPIK3CDTDO2ALDH1A1
SCHEMBL16848368 0.72 ALDH1A1 (0.46) PIK3CAPIK3CDPLAUHTR3EHTR3B
SCHEMBL989969 0.72 ASIC3 (0.51) PLAUHTR3EHTR3BHTR3ABACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118344355-A Quinazolinone derivative, preparation method thereof and application thereof in anti-inflammatory and anti-tumor 贵州省天然产物研究中心 2024-07-16 CN disclosed
CN-116253686-B Aminobenzimidazole benzamide derivative and application thereof 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) 2023-11-17 CN disclosed
CN-116253686-A Aminobenzimidazole benzamide derivative and application thereof 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) 2023-06-13 CN disclosed
CN-110655505-B 6- (2-amino-1H-benzo [ d ] imidazol-6-yl) quinazolin-4 (3H) -ones 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) 2022-06-21 CN disclosed