SCHEMBL29732889

SCHEMBL29732889

COC[C@H](C)Oc1nc2c(-c3cnn(C)c3)nc(-c3ccc(Cl)cc3)cn2n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 7/20 0.38
JAK1 P23458 7/20 0.38
TYK2 P29597 7/20 0.38
JAK3 P52333 7/20 0.38
F2RL3 Q96RI0 1/20 0.35
RET P07949 5/20 0.35
ALDH1A1 P00352 2/20 0.34
KCNH2 Q12809 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
HSD17B10 Q99714 1/20 0.34
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29498945 0.90 JAK2 (0.35) JAK2JAK1TYK2JAK3RET
SCHEMBL24539588 0.90 JAK2 (0.44) JAK2JAK1TYK2JAK3RET
SCHEMBL24539861 0.85 ALDH1A1 (0.39) JAK2JAK1TYK2JAK3F2RL3
SCHEMBL29732784 0.78 FGFR3 (0.44) JAK2JAK1TYK2JAK3F2RL3
SCHEMBL24539590 0.78 JAK2 (0.42) JAK2JAK1TYK2JAK3F2RL3
SCHEMBL24539461 0.78 JAK2 (0.42) JAK2JAK1TYK2JAK3F2RL3
SCHEMBL24539477 0.77 JAK2 (0.46) JAK2JAK1TYK2JAK3RET
SCHEMBL29733004 0.76 MAPT (0.42) JAK2JAK1TYK2JAK3F2RL3
SCHEMBL24327357 0.76 JAK2 (0.39) JAK2JAK1TYK2JAK3RET
SCHEMBL24539406 0.75 JAK2 (0.45) JAK2JAK1TYK2JAK3F2RL3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115698005-B Fused ring AhR inhibitors 山东轩竹医药科技有限公司 2024-02-06 CN disclosed
WO-2022127753-A1 FUSED RING AHR INHIBITOR 山东轩竹医药科技有限公司 2022-06-23 WO disclosed