SCHEMBL29732986

SCHEMBL29732986

CS(=O)(=O)c1ccc(-c2csc(=S)n2-c2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.58
PTGS1 P23219 2/20 0.54
CYP1A2 P05177 1/20 0.49
CYP2C19 P33261 1/20 0.49
CA12 O43570 4/20 0.47
CA1 P00915 4/20 0.47
CA2 P00918 4/20 0.47
CA9 Q16790 4/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5672477 0.86 CA12 (0.48) PTGS2PTGS1CA12CA1CA2
SCHEMBL5674063 0.86 PTGS2 (0.46) PTGS2PTGS1
SCHEMBL5674068 0.81 CA12 (0.62) PTGS2PTGS1CA12CA1CA2
SCHEMBL3831175 0.74 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL5672972 0.73 CA12 (0.60) PTGS2PTGS1CA12CA1CA2
SCHEMBL5671527 0.73 PTGS2 (0.56) PTGS2PTGS1CA12CA1CA2
SCHEMBL8076923 0.71 PTGS2 (0.61) PTGS2PTGS1CA12CA1CA2
SCHEMBL8397305 0.70 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL8303948 0.70 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL8071998 0.70 CA12 (0.63) PTGS2PTGS1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114634505-B Substituted indolone-chain-substituted-1, 3-thiazolidineone derivative and preparation method and application thereof 复旦大学 2024-05-24 CN disclosed
CN-114634506-B Substituted 1H-indol-2-one-yl-3, 5-substituted aryl-1, 3-thiazolidinedione derivatives 复旦大学 2024-04-19 CN disclosed
CN-114634505-A Substituted indolone-link-substituted-1, 3-thiazolidinone derivative and preparation method and application thereof 复旦大学 2022-06-17 CN disclosed
CN-114634506-A Substituted 1H-indol-2-one-link-3, 5-substituted aryl-1, 3-thiazolidinone derivatives 复旦大学 2022-06-17 CN disclosed