SCHEMBL29741063

SCHEMBL29741063

Oc1ccc2cnn(-c3cn[nH]c3)c2c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.43
HTR2C P28335 3/20 0.43
HTR2B P41595 3/20 0.43
LRRK2 Q5S007 3/20 0.41
HTR1A P08908 2/20 0.40
ADRA2A P08913 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
HTR1D P28221 1/20 0.40
HTR7 P34969 1/20 0.40
HTR4 Q13639 1/20 0.40
NR3C1 P04150 2/20 0.39
PGR P06401 1/20 0.36
CYP11B2 P19099 4/20 0.36
CYP11B1 P15538 2/20 0.36
KHK P50053 6/20 0.35
ERCC1 P07992 1/20 0.34
ERCC4 Q92889 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29539072 0.78 CYP11B2 (0.44) LRRK2ADRA2AADRA2BADRA2CNR3C1
Hydrochloric Acid SCHEMBL30557140 0.76 CYP11B2 (0.43) LRRK2ADRA2AADRA2BADRA2CNR3C1
SCHEMBL29493752 0.76 NR3C1 (0.62) HTR2AHTR2CHTR2BHTR1AADRA2A
SCHEMBL25368249 0.76 NR3C1 (0.62) HTR2AHTR2CHTR2BHTR1AADRA2A
SCHEMBL29741029 0.76 MAPT (0.43) LRRK2
SCHEMBL15505492 0.75 NR3C1 (0.65) HTR2AHTR2CHTR2BNR3C1PGR
SCHEMBL30557175 0.75 LRRK2 (0.37) LRRK2CYP11B2CYP11B1KHK
SCHEMBL29741008 0.73 HTR2A (0.47) HTR2AHTR2CHTR2BLRRK2HTR1A
SCHEMBL29539207 0.71 LRRK2 (0.33) LRRK2
SCHEMBL29741312 0.71 NR3C1 (0.42) HTR2AHTR2CHTR2BLRRK2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155419-A1 INDAZOLES AND AZAINDAZOLES AS LRRK2 INHIBITORS ESCAPE Bio, Inc. (US) 2022-07-21 WO disclosed