SCHEMBL29757378

SCHEMBL29757378

C=C(C)c1cccc(-c2ccnc(F)c2)c1CC(=O)OC.COC(=O)Cc1c(-c2ccnc(F)c2)cccc1C(C)C

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 6/20 0.36
ROCK1 Q13464 4/20 0.36
PRKACA P17612 3/20 0.36
PRKG1 Q13976 3/20 0.36
PRKACG P22612 2/20 0.36
PRKACB P22694 2/20 0.36
AKT1 P31749 2/20 0.36
CYP2C9 P11712 1/20 0.36
CYP3A4 P08684 2/20 0.35
DHODH Q02127 1/20 0.34
NLRP3 Q96P20 6/20 0.33
FFAR1 O14842 1/20 0.33
LPAR1 Q92633 2/20 0.32
MAPK1 P28482 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23012235 0.92 ROCK2 (0.40) ROCK2ROCK1PRKACAPRKG1PRKACG
SCHEMBL29691382 0.92 ROCK2 (0.40) ROCK2ROCK1PRKACAPRKG1PRKACG
SCHEMBL29691431 0.91 ROCK2 (0.41) ROCK2ROCK1PRKACAPRKG1PRKACG
SCHEMBL23012385 0.91 ROCK2 (0.41) ROCK2ROCK1PRKACAPRKG1PRKACG
SCHEMBL23013492 0.81 ROCK2 (0.45) ROCK2ROCK1PRKACAPRKG1PRKACG
SCHEMBL21962108 0.80 PKN1 (0.41) CYP3A4NLRP3
SCHEMBL23012645 0.79 CTSA (0.42) ROCK2ROCK1PRKACAPRKG1PRKACG
SCHEMBL29691436 0.79 CTSA (0.42) ROCK2ROCK1PRKACAPRKG1PRKACG
SCHEMBL21962081 0.79 NLRP3 (0.46) CYP3A4NLRP3LPAR1
SCHEMBL23012260 0.76 SMN1; SMN2 (0.44) ROCK2ROCK1PRKACAPRKG1PRKACG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4013762-A1 MACROCYCLIC SULFONYLAMIDE DERIVATIVES USEFUL AS NLRP3 INHIBITORS Inflazome Limited (IE) 2022-06-22 EP disclosed