SCHEMBL29757459

SCHEMBL29757459

CC(O)c1ccc(F)nc1Cl

nearest known ligand 0.41

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 2/20 0.41
KCNH2 Q12809 1/20 0.35
FFAR2 O15552 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23363400 1.00 PDE2A (0.41) PDE2AKCNH2FFAR2
SCHEMBL18368368 0.83 LMNA (0.33)
SCHEMBL25053869 0.79 PDE2A (0.42) PDE2AKCNH2
SCHEMBL3708356 0.79 PDE2A (0.39) PDE2AKCNH2
SCHEMBL3617710 0.79 PDE2A (0.35) PDE2A
SCHEMBL23363065 0.78 PDE2A (0.34) PDE2A
SCHEMBL23363064 0.78 PDE2A (0.34) PDE2A
SCHEMBL29757466 0.78 PDE2A (0.34) PDE2A
SCHEMBL31416770 0.76 PDE2A (0.37) PDE2A
SCHEMBL31416829 0.72 PDE2A (0.41) PDE2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115867556-B LPA receptor antagonists and uses thereof 吉利德科学公司 2025-05-06 CN disclosed
CN-114728168-B Triazole carbamate pyridylsulfonamides as LPA receptor antagonists and their use 吉利德科学公司 2024-04-09 CN disclosed
EP-4161641-A1 LPA RECEPTOR ANTAGONISTS AND USES THEREOF GILEAD SCIENCES, INC. (US) 2023-04-12 EP disclosed
EP-4161936-A1 LPA RECEPTOR ANTAGONISTS AND USES THEREOF GILEAD SCIENCES, INC. (US) 2023-04-12 EP disclosed
CN-115942972-A LPA receptor antagonists and uses thereof 吉利德科学公司 2023-04-07 CN disclosed
CN-115867556-A LPA receptor antagonists and uses thereof 吉利德科学公司 2023-03-28 CN disclosed
CN-114728168-A Triazolecarbamate pyridylsulfonamides as LPA receptor antagonists and their use 吉利德科学公司 2022-07-08 CN disclosed