SCHEMBL29775388

SCHEMBL29775388

COc1ccc(OC)c(-c2cccnc2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 10/20 0.61
CYP11B1 P15538 9/20 0.61
CYP17A1 P05093 5/20 0.60
CYP19A1 P11511 3/20 0.60
KDM4E B2RXH2 2/20 0.59
NPC1 O15118 2/20 0.59
NPSR1 Q6W5P4 1/20 0.59
CYP3A4 P08684 3/20 0.58
CYP1A2 P05177 2/20 0.56
CYP1A1 P04798 1/20 0.56
CYP1B1 Q16678 1/20 0.56
ALDH1A1 P00352 1/20 0.56
HPGD P15428 1/20 0.56
HSD17B10 Q99714 1/20 0.56
PDE4B Q07343 1/20 0.55
RAB9A P51151 1/20 0.55
HDAC4 P56524 1/20 0.55
HDAC2 Q92769 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
CYP2C9 P11712 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8165131 1.00 CYP11B2 (0.61) CYP11B2CYP11B1CYP17A1CYP19A1KDM4E
SCHEMBL14925557 0.84 CYP11B2 (0.74) CYP11B2CYP11B1CYP17A1CYP19A1KDM4E
SCHEMBL14003313 0.84 CYP11B1 (0.55) CYP11B2CYP11B1CYP17A1CYP19A1KDM4E
SCHEMBL1423147 0.83 KDM4E (0.69) CYP11B2CYP11B1CYP17A1CYP19A1KDM4E
SCHEMBL28118939 0.83 CYP11B1 (0.61) CYP11B2CYP11B1CYP17A1CYP19A1KDM4E
SCHEMBL2652791 0.83 MKNK1 (0.55) CYP11B2CYP11B1CYP17A1CYP19A1KDM4E
SCHEMBL6217515 0.83 CYP11B1 (0.54) CYP11B2CYP11B1CYP17A1CYP19A1KDM4E
SCHEMBL28225240 0.81 MKNK1 (0.60) CYP11B2CYP11B1CYP17A1CYP19A1KDM4E
SCHEMBL8502557 0.81 CYP17A1 (0.55) CYP11B2CYP11B1CYP17A1KDM4ENPC1
SCHEMBL7372635 0.81 CYP11B2 (0.52) CYP11B2CYP11B1CYP17A1CYP19A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114761083-B 5-HT for treating depression 2A Agonists 罗福拉公司 2024-02-13 CN disclosed
CN-114761083-A 5-HT for the treatment of depression2AAgonists 罗福拉公司 2022-07-15 CN disclosed